WDR5-IN-6（Cat No.:I041058）is a small molecule inhibitor targeting WDR5 (WD repeat domain 5), a key protein involved in the regulation of gene expression through its interaction with histone methyltransferase complexes. By disrupting the WDR5-MLL (mixed-lineage leukemia)

WDR5-IN-6 is a WDR5 inhibitor, targeting to WBM site. WDR5-IN-6 inhibits cell proliferation of neuroblastoma cell lines with potent anti-tumor activity. WDR5-IN-6 shows high synergy with OICR-9429 (HY-16993), a WDR5 inhibitor targeting to WIN site.